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Identification and pharmacological characterization of cholesterol-5,6-epoxide hydrolase as a target for tamoxifen and AEBS ligands

The microsomal antiestrogen binding site (AEBS) is a high-affinity target for the antitumor drug tamoxifen and its cognate ligands that mediate breast cancer cell differentiation and apoptosis. The AEBS, a hetero-oligomeric complex composed of 3β-hydroxysterol-Δ(8)-Δ(7)-isomerase (D8D7I) and 3β-hydr...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: de Medina, Philippe, Paillasse, Michael R., Segala, Gregory, Poirot, Marc, Silvente-Poirot, Sandrine
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: National Academy of Sciences 2010
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2922168/
https://ncbi.nlm.nih.gov/pubmed/20615952
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1002922107
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