Caricamento...

Insights in 17β-HSD1 Enzyme Kinetics and Ligand Binding by Dynamic Motion Investigation

BACKGROUND: Bisubstrate enzymes, such as 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1), exist in solution as an ensemble of conformations. 17β-HSD1 catalyzes the last step of the biosynthesis of estradiol and, thus, it is a potentially attractive target for breast cancer treatment. METHODOLOGY/...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Negri, Matthias, Recanatini, Maurizio, Hartmann, Rolf W.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2010
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2919385/
https://ncbi.nlm.nih.gov/pubmed/20706575
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0012026
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !