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The Structure-Activity Relationships of A-Ring-Substituted Aromathecin Topoisomerase I Inhibitors Strongly Support a Camptothecin-Like Binding Mode

Aromathecins are inhibitors of human topoisomerase I (Top1). These compounds are composites of several heteroaromatic systems, namely the camptothecins and indenoisoquinolines, and they possess notable Top1 inhibition and cytotoxicity when substituted at position 14. The SAR of these compounds overl...

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Detalhes bibliográficos
Main Authors: Cinelli, Maris A., Morrell, Andrew E., Dexheimer, Thomas S., Agama, Keli, Agrawal, Surbhi, Pommier, Yves, Cushman, Mark
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2911012/
https://ncbi.nlm.nih.gov/pubmed/20630766
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2010.06.040
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