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Broad Spectrum Alkynyl Inhibitors of T315I Bcr-Abl

A series of alkyne containing type II inhibitors with potent inhibitory activity of T315I Bcr-Abl has been identified. The most active compound 4 exhibits an EC(50) of less than 1 nM against wild-type Bcr-Abl and an EC(50) of 10 nM against T315I mutant but is broadly active against a number of other...

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Hlavní autoři: Deng, Xianming, Lim, Sang Min, Zhang, Jianming, Gray, Nathanael S.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2010
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2901992/
https://ncbi.nlm.nih.gov/pubmed/20541934
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2010.05.043
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