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Convergent synthesis of α-ketoamide inhibitors of Pin1

[Image: see text] A convergent synthesis of α-ketoamide inhibitors of Pin1 is described. An α-hydroxyorthothioester derivative of Ser was reacted directly with an amine synthon. The reaction was catalyzed by HgO and HgCl(2) to form α-hydroxyamide. Thus, hydrolysis and coupling were combined in one s...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Xu, Guoyan G., Etzkorn, Felicia A.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2010
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC2844255/
https://ncbi.nlm.nih.gov/pubmed/20102178
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol9027013
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