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Gold(I)-Catalyzed Intramolecular Dihydroamination of Allenes with N,N′-Disubstituted Ureas to Form Bicyclic Imidazolidin-2-ones

[Image: see text] Reaction of N-δ-allenyl urea 1 with a catalytic 1:1 mixture of gold(I) N-heterocyclic carbene complex (5)AuCl [5 = 1,3-bis(2,6-diisopropylphenyl)imidazol-2-ylidine] and AgPF(6) at room temperature for 2 h led to isolation of bicyclic imidazolidin-2-one 4 in 93% yield as a single di...

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Detalhes bibliográficos
Main Authors: Li, Hao, Widenhoefer, Ross A.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2813268/
https://ncbi.nlm.nih.gov/pubmed/19514795
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol900730w
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