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Inhibitors of the Mitochondrial Citrate Transport Protein: Validation of the Role of Substrate Binding Residues and Discovery of the First Purely Competitive Inhibitor

The mitochondrial citrate transport protein (CTP) is critical to energy metabolism in eukaryotic cells. We demonstrate that 1,2,3-benzenetricarboxylate (BTC), the classic and defining inhibitor of the mitochondrial CTP, is a mixed inhibitor of the reconstituted Cys-less CTP, with a strong competitiv...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Aluvila, Sreevidya, Sun, Jiakang, Harrison, David H. T., Walters, D. Eric, Kaplan, Ronald S.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: The American Society for Pharmacology and Experimental Therapeutics 2010
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2802432/
https://ncbi.nlm.nih.gov/pubmed/19843634
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.109.058750
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