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Inhibitors of the Mitochondrial Citrate Transport Protein: Validation of the Role of Substrate Binding Residues and Discovery of the First Purely Competitive Inhibitor

The mitochondrial citrate transport protein (CTP) is critical to energy metabolism in eukaryotic cells. We demonstrate that 1,2,3-benzenetricarboxylate (BTC), the classic and defining inhibitor of the mitochondrial CTP, is a mixed inhibitor of the reconstituted Cys-less CTP, with a strong competitiv...

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Detalhes bibliográficos
Main Authors: Aluvila, Sreevidya, Sun, Jiakang, Harrison, David H. T., Walters, D. Eric, Kaplan, Ronald S.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2802432/
https://ncbi.nlm.nih.gov/pubmed/19843634
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.109.058750
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