載入...

Discovery and SAR of 6-substituted-4-anilinoquinazolines as non-competitive antagonists of mGlu(5)

A high-throughput cell-based screen identified a series of 6-substituted-4-anilinoquinazolines as non-competitive antagonists of metabotropic glutamate receptor 5 (mGlu(5)). This communication describes the SAR of this series and the profile of selected compounds in selectivity and radioligand bindi...

全面介紹

Na minha lista:
書目詳細資料
Main Authors: Felts, Andrew S., Saleh, Sam A., Le, Uyen, Rodriguez, Alice L., Weaver, C. David, Conn, P. Jeffrey, Lindsley, Craig W., Emmitte, Kyle A.
格式: Artigo
語言:Inglês
出版: 2009
主題:
在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC2801349/
https://ncbi.nlm.nih.gov/pubmed/19854049
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2009.10.024
標簽: 添加標簽
沒有標簽, 成為第一個標記此記錄!