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SB265610 is an allosteric, inverse agonist at the human CXCR2 receptor

BACKGROUND AND PURPOSE: In several previous studies, the C-X-C chemokine receptor (CXCR)2 antagonist 1-(2-bromo-phenyl)-3-(7-cyano-3H-benzotriazol-4-yl)-urea (SB265610) has been described as binding competitively with the endogenous agonist. This is in contrast to many other chemokine receptor antag...

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Detalles Bibliográficos
Autores principales: Bradley, ME, Bond, ME, Manini, J, Brown, Z, Charlton, SJ
Formato: Artigo
Lenguaje:Inglês
Publicado: Blackwell Publishing Ltd 2009
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2795238/
https://ncbi.nlm.nih.gov/pubmed/19422399
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2009.00182.x
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