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Studies Toward the Pharmacophore of Salvinorin A, a Potent Kappa Opioid Receptor Agonist

Salvinorin A (1), from the sage Salvia divinorum, is a potent and selective kappa opioid receptor (KOR) agonist. We screened other salvinorins and derivatives for binding affinity and functional activity at opioid receptors. Our results suggest that the methyl ester and furan ring are required for a...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Munro, Thomas A., Rizzacasa, Mark A., Roth, Bryan L., Toth, Beth A., Yan, Feng
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2005
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2777653/
https://ncbi.nlm.nih.gov/pubmed/15658846
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm049438q
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