A carregar...

Inhibition of drug metabolizing cytochrome P450s by the aromatase inhibitor drug letrozole and its major oxidative metabolite 4,4′-methanol-bisbenzonitrile in vitro

PURPOSE: To determine the inhibitory potency of letrozole and its main human metabolite, 4,4′-methanol-bisbenzonitrilee, on the activities of eight cytochrome P450 (CYP) enzymes. METHODS: Letrozole and its metabolite were incubated with human liver microsomes (HLMs) (or expressed CYP isoforms) and N...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Jeong, Seongwook, Woo, Margaret M., Flockhart, David A., Desta, Zeruesenay
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2774495/
https://ncbi.nlm.nih.gov/pubmed/19198839
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00280-009-0935-7
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!