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Insight to pyrazinamide resistance inMycobacterium tuberculosisby molecular docking

Pyrazinamide (PZA) - an important drug in the anti-tuberculosis therapy, activated by an enzyme Pyrazinamidase (PZase). The basis of PZA resistance in Mycobacterium tuberculosis was owing to mutation in pncA gene coding for PZase. Homology modeling of PZase was performed using software Discovery Stu...

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Библиографические подробности
Главные авторы: Unissa, Amirudeen Nusrath, Selvakumar, Nagamiah, Hassan, Sameer
Формат: Artigo
Язык:Inglês
Опубликовано: Biomedical Informatics 2009
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2770367/
https://ncbi.nlm.nih.gov/pubmed/20011149
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