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Insight to pyrazinamide resistance inMycobacterium tuberculosisby molecular docking

Pyrazinamide (PZA) - an important drug in the anti-tuberculosis therapy, activated by an enzyme Pyrazinamidase (PZase). The basis of PZA resistance in Mycobacterium tuberculosis was owing to mutation in pncA gene coding for PZase. Homology modeling of PZase was performed using software Discovery Stu...

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Detalhes bibliográficos
Main Authors: Unissa, Amirudeen Nusrath, Selvakumar, Nagamiah, Hassan, Sameer
Formato: Artigo
Idioma:Inglês
Publicado em: Biomedical Informatics 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2770367/
https://ncbi.nlm.nih.gov/pubmed/20011149
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