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The Pneumotoxin 3-Methylindole Is a Substrate and a Mechanism-Based Inactivator of CYP2A13, a Human Cytochrome P450 Enzyme Preferentially Expressed in the Respiratory Tract

3-Methylindole (3MI), a respiratory tract toxicant, can be metabolized by a number of cytochromes P450 (P450), primarily through either dehydrogenation or epoxidation of the indole. In the present study, we assessed the bioactivation of 3MI by recombinant CYP2A13, a human P450 predominantly expresse...

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Bibliografske podrobnosti
Main Authors: D'Agostino, Jaime, Zhuo, Xiaoliang, Shadid, Mohammad, Morgan, Daniel G., Zhang, Xiuling, Humphreys, W. Griffith, Shu, Yue-Zhong, Yost, Garold S., Ding, Xinxin
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2009
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2769036/
https://ncbi.nlm.nih.gov/pubmed/19608696
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.109.027300
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