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Discovery and Development of a Small Molecule Library with Lumazine Synthase Inhibitory Activity

(E)-5-Nitro-6-(2-hydroxystyryl)pyrimidine-2,4(1H,3H)-dione (9) was identified as a novel inhibitor of Schizosaccharomyces pombe lumazine synthase by high-throughput screening of a 100,000 compound library. The K(i) of 9 vs. Mycobacterium tuberculosis lumazine synthase was 95 μM. Compound 9 is a stru...

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Autors principals: Talukdar, Arindam, Breen, Megan, Bacher, Adelbert, Illarionov, Boris, Fischer, Markus, Georg, Gunda, Ye, Qi-Zhuang, Cushman, Mark
Format: Artigo
Idioma:Inglês
Publicat: 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2760403/
https://ncbi.nlm.nih.gov/pubmed/19552377
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jo900238q
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