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The Nucleoside Analog D-carba T Blocks HIV-1 Reverse Transcription

A major pathway for HIV-1 resistance to nucleoside reverse transcriptase inhibitors (NRTIs) involves reverse transcriptase (RT) mutations that enhance ATP-dependent pyrophosphorolysis, which excises NRTIs from the end of viral DNA. We analyzed novel NRTIs for their ability to inhibit DNA synthesis o...

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Autors principals: Boyer, Paul L., Vu, B. Christie, Ambrose, Zandrea, Julias, John G., Warnecke, Svenja, Liao, Chenzhong, Meier, Chris, Marquez, Victor E., Hughes, Stephen H.
Format: Artigo
Idioma:Inglês
Publicat: 2009
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2756836/
https://ncbi.nlm.nih.gov/pubmed/19678643
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm801176e
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