Nalaganje...

Molecular modeling of G-protein coupled receptor kinase 2: Docking and biochemical evaluation of inhibitors

G-protein coupled receptor kinase 2 (GRK2) regulates the activity of many receptors. Because potent inhibitors of GRK2 are thus far limited to polyanionic compounds like heparin, we searched for new inhibitors with the aid of a molecular model of GRK2. We used the available crystal structure of cAMP...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
Main Authors: Kassack, Matthias U., Högger, Petra, Gschwend, Daniel A., Kameyama, Kimihiko, Haga, Tatsuya, Graul, Richard C., Sadée, Wolfgang
Format: Artigo
Jezik:Inglês
Izdano: Springer-Verlag 2000
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2750997/
https://ncbi.nlm.nih.gov/pubmed/11741218
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/ps020102
Oznake: Označite
Brez oznak, prvi označite!