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Molecular modeling of G-protein coupled receptor kinase 2: Docking and biochemical evaluation of inhibitors

G-protein coupled receptor kinase 2 (GRK2) regulates the activity of many receptors. Because potent inhibitors of GRK2 are thus far limited to polyanionic compounds like heparin, we searched for new inhibitors with the aid of a molecular model of GRK2. We used the available crystal structure of cAMP...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Päätekijät: Kassack, Matthias U., Högger, Petra, Gschwend, Daniel A., Kameyama, Kimihiko, Haga, Tatsuya, Graul, Richard C., Sadée, Wolfgang
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Springer-Verlag 2000
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC2750997/
https://ncbi.nlm.nih.gov/pubmed/11741218
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/ps020102
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