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Genetic variations in human G protein-coupled receptors: Implications for drug therapy

Numerous genes encode G protein-coupled receptors (GPCRs)-a main molecular target for drug therapy. Estimates indicate that the human genome contains approximately 600 GPCR genes. This article addresses therapeutic implications of sequence variations in GPCR genes. A number of inactivating and activ...

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Autori principali: Sadee, Wolfgang, Hoeg, Elen, Lucas, Julie, Wang, Danxin
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer-Verlag 2001
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2751017/
https://ncbi.nlm.nih.gov/pubmed/11741273
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/ps030322
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