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Identification of Quinolines that Inhibit Melanogenesis by Altering Tyrosinase Family Trafficking

A series of quinolines, including chloroquine and quinine, were identified as potent pigmentation inhibitors through screening a compound library in murine melanocytes. Structure-activity relationship analysis indicated that 4-substituted amino groups with a tertiary amine side chain, such as chloro...

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Autors principals: Ni-Komatsu, Li, Tong, ChunXiang, Chen, Guangming, Brindzei, Nelya, Orlow, Seth J.
Format: Artigo
Idioma:Inglês
Publicat: 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2747315/
https://ncbi.nlm.nih.gov/pubmed/18801917
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.108.050633
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