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AFN-1252, a FabI Inhibitor, Demonstrates a Staphylococcus-Specific Spectrum of Activity

AFN-1252, a potent inhibitor of enoyl-acyl carrier protein reductase (FabI), inhibited all clinical isolates of Staphylococcus aureus (n = 502) and Staphylococcus epidermidis (n = 51) tested, including methicillin (meticillin)-resistant isolates, at concentrations of ≤0.12 μg/ml. In contrast, AFN-12...

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Auteurs principaux: Karlowsky, James A., Kaplan, Nachum, Hafkin, Barry, Hoban, Daryl J., Zhanel, George G.
Format: Artigo
Langue:Inglês
Publié: American Society for Microbiology (ASM) 2009
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Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2715641/
https://ncbi.nlm.nih.gov/pubmed/19487444
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00400-09
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