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Analogs of the marine alkaloid makaluvamines: Synthesis, topoisomerase II inhibition and anticancer activity

Twelve analogs of makaluvamines have been synthesized. These compounds were evaluated for their ability to inhibit the enzyme topoisomerase II. Five compounds were shown to inhibit topoisomerase catalytic activity comparable to two known topoisomerase II targeting control drugs, etoposide and m-AMSA...

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Autori principali: Shinkre, Bidhan A., Raisch, Kevin P., Fan, Liming, Velu, Sadanandan E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2007
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2706148/
https://ncbi.nlm.nih.gov/pubmed/17368022
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2007.02.065
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