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Analogs of the marine alkaloid makaluvamines: Synthesis, topoisomerase II inhibition and anticancer activity

Twelve analogs of makaluvamines have been synthesized. These compounds were evaluated for their ability to inhibit the enzyme topoisomerase II. Five compounds were shown to inhibit topoisomerase catalytic activity comparable to two known topoisomerase II targeting control drugs, etoposide and m-AMSA...

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Détails bibliographiques
Auteurs principaux: Shinkre, Bidhan A., Raisch, Kevin P., Fan, Liming, Velu, Sadanandan E.
Format: Artigo
Langue:Inglês
Publié: 2007
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2706148/
https://ncbi.nlm.nih.gov/pubmed/17368022
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2007.02.065
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