Loading...

Mutations of the GABA-A receptor α1 subunit M1 domain reveal unexpected complexity for modulation by neuroactive steroids

Neuroactive steroids are among the most efficacious modulators of the mammalian GABA-A receptor. Previous work has proposed that receptor potentiation is mediated by steroid interactions with a site defined by the residues α1N407/Y410 in the M4 transmembrane domain, and residue α1Q241 in the M1 doma...

Full description

Saved in:
Bibliographic Details
Main Authors: Akk, Gustav, Li, Ping, Bracamontes, John, Reichert, David E., Covey, Douglas F., Steinbach, Joe Henry
Format: Artigo
Language:Inglês
Published: 2008
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC2701692/
https://ncbi.nlm.nih.gov/pubmed/18544665
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.108.048520
Tags: Add Tag
No Tags, Be the first to tag this record!