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Anti-tumor Compounds Based on a Natural Product Consensus Pharmacophore

We report the design and highly enantioselective synthesis of a potent analog of the spliceosome inhibitor FR901464, based on a non-natural product scaffold. The design of this compound was facilitated by a pharmacophore hypothesis that assumed key interaction types that are common to FR901464 and a...

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Autori principali: Lagisetti, Chandraiah, Pourpak, Alan, Jiang, Qin, Cui, Xiaoli, Goronga, Tinopiwa, Morris, Stephan W., Webb, Thomas R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2008
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2701350/
https://ncbi.nlm.nih.gov/pubmed/18788726
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm8006195
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