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Analysis of Full and Partial Agonists Binding to β(2)-Adrenergic Receptor Suggests a Role of Transmembrane Helix V in Agonist-Specific Conformational Changes

The 2.4 Å crystal structure of the β(2)-adrenergic receptor (β(2)AR) in complex with the high-affinity inverse agonist (-)-carazolol provides a detailed structural framework for the analysis of ligand recognition by adrenergic receptors. Insights into agonist binding and the corresponding conformati...

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Bibliografski detalji
Glavni autori: Katritch, Vsevolod, Reynolds, Kimberly A., Cherezov, Vadim, Hanson, Michael A., Roth, Christopher B., Yeager, Mark, Abagyan, Ruben
Format: Artigo
Jezik:Inglês
Izdano: 2009
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2693451/
https://ncbi.nlm.nih.gov/pubmed/19353579
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jmr.949
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