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Effect of Pluronic P85 on ATPase Activity of Drug Efflux Transporters

PURPOSE: Pluronic block copolymers are potent sensitizers of multi-drug resistant (MDR) cancer cells. The sensitization effect by Pluronics is a result of two processes acting in concert: i) intracellular ATP depletion, and ii) inhibition of ATPase activity of drug efflux proteins. This work charact...

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Detalhes bibliográficos
Main Authors: Batrakova, Elena V., Li, Shu, Li, Yili, Alakhov, Valery Yu., Kabanov, Alexander V.
Formato: Artigo
Idioma:Inglês
Publicado em: 2004
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2677181/
https://ncbi.nlm.nih.gov/pubmed/15648254
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