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Activation of ATR and related PIKKs

The DNA damage response kinase ATR is an essential regulator of genome integrity. TopBP1 functions as a general activator of ATR. We have recently shown that TopBP1 activates ATR through its regulatory subunit ATRIP and a PIKK regulatory domain (PRD) located adjacent to its kinase domain. This mecha...

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Detalles Bibliográficos
Main Authors: Mordes, Daniel A., Cortez, David
Formato: Artigo
Idioma:Inglês
Publicado: 2008
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2672405/
https://ncbi.nlm.nih.gov/pubmed/18769153
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