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The second transmembrane domain of the large conductance, voltage- and calcium-gated potassium channel β(1) subunit is a lithocholate sensor

Bile acids and other steroids modify BK channel activity contributing to nongenomic modulation of myogenic tone. The protein regions that sense steroid action, however, remain unknown. Accessory BK β(1) subunits are necessary for lithocholate to activate BK channels and vasodilate. Using recombinant...

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Autors principals: Bukiya, Anna N., Vaithianathan, Thirumalini, Toro, Ligia, Dopico, Alejandro M.
Format: Artigo
Idioma:Inglês
Publicat: 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2665905/
https://ncbi.nlm.nih.gov/pubmed/18242174
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.febslet.2008.01.036
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