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A small molecule inhibitor 1,2,4,5-Benzenetetraamine tetrahydrochloride, targeting the Y397 site of Focal Adhesion Kinase decreases tumor growth

Focal Adhesion Kinase (FAK) is a non-receptor kinase that is overexpressed in many types of tumors. We developed a novel cancer-therapy approach, targeting the main autophosphorylation site of FAK, Y397 by computer modeling and screening of the National Cancer Institute (NCI) small molecule compound...

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Библиографические подробности
Главные авторы: Golubovskaya, Vita M., Nyberg, Carl, Zheng, Min, Kweh, Frederick, Magis, Andrew, Ostrov, David, Cance, William G.
Формат: Artigo
Язык:Inglês
Опубликовано: 2008
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2662449/
https://ncbi.nlm.nih.gov/pubmed/18989950
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm800483v
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