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Raltegravir, elvitegravir, and metoogravir: the birth of "me-too" HIV-1 integrase inhibitors

Merck's MK-0518, known as raltegravir, has recently become the first FDA-approved HIV-1 integrase (IN) inhibitor and has since risen to blockbuster drug status. Much research has in turn been conducted over the last few years aimed at recreating but optimizing the compound's interactions w...

Täydet tiedot

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Bibliografiset tiedot
Päätekijät: Serrao, Erik, Odde, Srinivas, Ramkumar, Kavya, Neamati, Nouri
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: BioMed Central 2009
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC2660292/
https://ncbi.nlm.nih.gov/pubmed/19265512
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1742-4690-6-25
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