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Biochemical, Functional, and Pharmacological Characterization of AT-56, an Orally Active and Selective Inhibitor of Lipocalin-type Prostaglandin D Synthase

We report here that 4-dibenzo[a,d]cyclohepten-5-ylidene-1-[4-(2H-tetrazol-5-yl)-butyl]-piperidine (AT-56) is an orally active and selective inhibitor of lipocalin-type prostaglandin (PG) D synthase (L-PGDS). AT-56 inhibited human and mouse L-PGDSs in a concentration (3–250 μm)-dependent manner but d...

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Autors principals: Irikura, Daisuke, Aritake, Kosuke, Nagata, Nanae, Maruyama, Toshihiko, Shimamoto, Shigeru, Urade, Yoshihiro
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2658056/
https://ncbi.nlm.nih.gov/pubmed/19131342
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M808593200
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