A carregar...

Synthesis and Biological Evaluation of a Novel Pentagastrin-Toxin Conjugate Designed for a Targeted Prodrug Mono-therapy of Cancer

A novel carbamate prodrug 2 containing a pentagastrin moiety was synthesized. 2 was designed as a detoxified analogue of the highly cytotoxic natural antibiotic duocarmycin SA (1) for the use in a targeted prodrug monotherapy of cancers expressing cholecystokinin (CCK-B)/gastrin receptors. The synth...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Tietze, Lutz F., Panknin, Olaf, Krewer, Birgit, Major, Felix, Schuberth, Ingrid
Formato: Artigo
Idioma:Inglês
Publicado em: Molecular Diversity Preservation International (MDPI) 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2635707/
https://ncbi.nlm.nih.gov/pubmed/19325786
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms9050821
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!