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Cisplatin Abrogates the Geldanamycin-induced Heat Shock Response

Benzoquinone ansamycin antibiotics such as geldanamycin (GA) bind to the N-terminal ATP binding domain of Hsp90 and inhibit its chaperone functions. Despite in vitro and in vivo studies indicating promising antitumor activity, derivatives of GA, including 17-AAG have demonstrated little clinical eff...

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Autors principals: McCollum, Andrea K., Lukasiewicz, Kara B., TenEyck, Cynthia J., Lingle, Wilma L., Toft, David O., Erlichman, Charles
Format: Artigo
Idioma:Inglês
Publicat: 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2572571/
https://ncbi.nlm.nih.gov/pubmed/18852129
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-08-0157
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