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Effects of High-Affinity Inhibitors on Partial Reactions, Charge Movements, and Conformational States of the Ca(2+) Transport ATPase (Sarco-Endoplasmic Reticulum Ca(2+) ATPase)
The inhibitory effects of thapsigargin, cyclopiazonic acid, and 2,5-di(tert-butyl)hydroquinone, and 1,3-dibromo-2,4,6-tri(methylisothiouronium)benzene on the Ca(2+) ATPase were characterized by comparative measurements of sequential reactions of the catalytic and transport cycle, including biochemic...
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| Autores principales: | , , , , , |
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| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
2008
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| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2564850/ https://ncbi.nlm.nih.gov/pubmed/18212248 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.107.043745 |
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