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The Peripheral Benzodiazepine Receptor Ligand 1-(2-Chlorophenyl-methylpropyl)-3-isoquinoline-carboxamide Is a Novel Antagonist of Human Constitutive Androstane Receptor

As a promiscuous xenobiotic sensor, the constitutive androstane receptor (CAR; NR1I3) regulates the expression of multiple drug metabolizing enzymes and transporters in liver. The constitutively activated nature of CAR in the cell-based transfection assays has hindered its utilization as a predictor...

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Autores principales: Li, Linhao, Chen, Tao, Stanton, Joseph D, Sueyoshi, Tatsuya, Negishi, Masahiko, Wang, Hongbing
Formato: Artigo
Lenguaje:Inglês
Publicado: 2008
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2562670/
https://ncbi.nlm.nih.gov/pubmed/18492798
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.108.046656
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