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Modifications of human carboxylesterase for improved prodrug activation

BACKGROUND: Carboxylesterases (CE) are ubiquitous enzymes responsible for the hydrolysis of numerous clinically useful drugs. Since ester moieties are frequently included in molecules to improve their water solubility and bioavailability, de facto they become substrates for CEs. OBJECTIVE: In this r...

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Detalhes bibliográficos
Main Authors: Hatfield, M. Jason, Wierdl, Monika, Wadkins, Randy M., Potter, Philip M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2556898/
https://ncbi.nlm.nih.gov/pubmed/18721110
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/17425255.4.9.1153
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