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Synthesis and Structure-Activity Relationships of Linear and Conformationally Constrained Peptide Analogs of CIYKYY as Src Tyrosine Kinase Inhibitors
A series of peptide analogs of Ac-CIYKYY (1) were synthesized by functional group modifications in peptide side chains or introducing conformational constraints, to improve the inhibitory potency against active Src kinase. Ac-CIYKF(4-NO(2))Y (2, IC(50) = 0.53 μM) and the conformationally constrained...
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| Main Authors: | , , , , , |
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| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
2006
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2527579/ https://ncbi.nlm.nih.gov/pubmed/16722659 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm060334k |
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