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Some Effects of CB1 Antagonists with Inverse Agonist and Neutral Biochemical Properties,

The CB1 inverse agonist/antagonist SR141716A recently has been introduced for the management of obesity (rimonabant; Acomplia) and appears to have beneficial effects. However, its utility may be hampered in some individuals by adverse effects including nausea or emesis or by mood depression. The rec...

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Autors principals: Bergman, Jack, Delatte, Marcus. S., Paronis, Carol A., Vemuri, Kiran, Pandarinathan, Pathi, Thakur, Ganesh A., Makriyannis, Alex
Format: Artigo
Idioma:Inglês
Publicat: 2007
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2441972/
https://ncbi.nlm.nih.gov/pubmed/18076956
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.physbeh.2007.11.007
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