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The kinetics of competitive antagonism of nicotinic acetylcholine receptors at physiological temperature

Detailed information about the ligand-binding site of nicotinic acetylcholine receptors has emerged from structural and mutagenesis experiments. However, these approaches provide only static images of ligand–receptor interactions. Kinetic measurements of changes in protein function are needed to dev...

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Autores principales: Demazumder, Deeptankar, Dilger, James P
Formato: Artigo
Lenguaje:Inglês
Publicado: Blackwell Science Inc 2008
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2375649/
https://ncbi.nlm.nih.gov/pubmed/18063662
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1113/jphysiol.2007.143289
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