Chargement en cours...

High-resolution crystal structures of ribonuclease A complexed with adenylic and uridylic nucleotide inhibitors. Implications for structure-based design of ribonucleolytic inhibitors

The crystal structures of bovine pancreatic ribonuclease A (RNase A) in complex with 3′,5′-ADP, 2′,5′-ADP, 5′-ADP, U-2′-p and U-3′-p have been determined at high resolution. The structures reveal that each inhibitor binds differently in the RNase A active site by anchoring a phosphate group in subsi...

Description complète

Enregistré dans:
Détails bibliographiques
Auteurs principaux: Leonidas, Demetres D., Chavali, Gayatri B., Oikonomakos, Nikos G., Chrysina, Evangelia D., Kosmopoulou, Magda N., Vlassi, Metaxia, Frankling, Claire, Acharya, K. Ravi
Format: Artigo
Langue:Inglês
Publié: Cold Spring Harbor Laboratory Press 2003
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2366950/
https://ncbi.nlm.nih.gov/pubmed/14573867
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!