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Clinical experience with the novel histone deacetylase inhibitor vorinostat (suberoylanilide hydroxamic acid) in patients with relapsed lymphoma

Preclinical studies indicate that vorinostat (suberoylanilide hydroxamic acid or SAHA) inhibits histone deacetylase (HDAC) activity, increases acetylated histones H2a, H2b, H3, and H4, and thereby induces differentiation and apoptosis in a variety of tumour cell lines, including murine erythroleukae...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखक: O'Connor, O A
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: Nature Publishing Group 2006
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC2360773/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjc.6603464
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