A carregar...

Induced-fit or preexisting equilibrium dynamics? Lessons from protein crystallography and MD simulations on acetylcholinesterase and implications for structure-based drug design

Crystal structures of acetylcholinesterase complexed with ligands are compared with side-chain conformations accessed by native acetylcholinesterase in molecular dynamics (MD) simulations. Several crystallographic conformations of a key residue in a specific binding site are accessed in a simulation...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Xu, Yechun, Colletier, Jacques Ph., Jiang, Hualiang, Silman, Israel, Sussman, Joel L., Weik, Martin
Formato: Artigo
Idioma:Inglês
Publicado em: Cold Spring Harbor Laboratory Press 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2271175/
https://ncbi.nlm.nih.gov/pubmed/18359854
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1110/ps.083453808
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!