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Design, Synthesis, and Evaluation of 10-N-Substituted Acridones as Novel Chemosensitizers in Plasmodium falciparum

A series of novel 10-N-substituted acridones, bearing alkyl side chains with tertiary amine groups at the terminal position, were designed, synthesized, and evaluated for the ability to enhance the potency of quinoline drugs against multidrug-resistant (MDR) Plasmodium falciparum malaria parasites....

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Kelly, Jane X., Smilkstein, Martin J., Cooper, Roland A., Lane, Kristin D., Johnson, Robert A., Janowsky, Aaron, Dodean, Rozalia A., Hinrichs, David J., Winter, Rolf, Riscoe, Michael
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Society for Microbiology (ASM) 2007
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2151415/
https://ncbi.nlm.nih.gov/pubmed/17846138
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00669-07
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