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Charge at the lidocaine binding site residue Phe-1759 affects permeation in human cardiac voltage-gated sodium channels

Our homology molecular model of the open/inactivated state of the Na(+) channel pore predicts, based on extensive mutagenesis data, that the local anaesthetic lidocaine docks eccentrically below the selectivity filter, such that physical occlusion is incomplete. Electrostatic field calculations sugg...

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Autors principals: McNulty, Megan M, Edgerton, Gabrielle B, Shah, Ravi D, Hanck, Dorothy A, Fozzard, Harry A, Lipkind, Gregory M
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Science Inc 2007
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2075178/
https://ncbi.nlm.nih.gov/pubmed/17363383
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1113/jphysiol.2007.130161
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