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Effects of clarithromycin and grapefruit juice on the pharmacokinetics of glibenclamide

WHAT IS ALREADY KNOWN ABOUT THIS SUBJECT: Severe hypoglycaemia has been reported after concomitant use of clarithromycin and glibenclamide. Glibenclamide is a substrate for the transporters P-glycoprotein and OATP2B1. Clarithromycin inhibits P-glycoprotein and grapefruit juice inhibits OATP2B1. WHAT...

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Autors principals: Lilja, Jari J, Niemi, Mikko, Fredrikson, Hanna, Neuvonen, Pertti J
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Science Inc 2007
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2000598/
https://ncbi.nlm.nih.gov/pubmed/17223855
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1365-2125.2006.02836.x
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