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Pharmacological specificity of novel, synthetic, cyclic peptides as antagonists at tachykinin receptors.

1. The interaction at tachykinin receptors of a series of novel cyclic hexapeptides has been examined by use of radioligand binding assays (NK1 and NK3 sites in rat cortex, NK2 sites in hamster urinary bladder) and functional pharmacological assays (guinea-pig ileum, rat vas deferens and rat portal...

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Main Authors: McKnight, A. T., Maguire, J. J., Elliott, N. J., Fletcher, A. E., Foster, A. C., Tridgett, R., Williams, B. J., Longmore, J., Iversen, L. L.
Formato: Artigo
Idioma:Inglês
Publicado: 1991
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC1908569/
https://ncbi.nlm.nih.gov/pubmed/1665732
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