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Structural basis for stem cell factor–KIT signaling and activation of class III receptor tyrosine kinases

Stem cell factor (SCF) binds to and activates the KIT receptor, a class III receptor tyrosine kinase (RTK), to stimulate diverse processes including melanogenesis, gametogenesis and hematopoeisis. Dysregulation of KIT activation is associated with many cancers. We report a 2.5 Å crystal structure of...

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Détails bibliographiques
Auteurs principaux: Liu, Heli, Chen, Xiaoyan, Focia, Pamela J, He, Xiaolin
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group 2007
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC1794399/
https://ncbi.nlm.nih.gov/pubmed/17255936
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.emboj.7601545
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