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Modulation of P-glycoprotein activity by cannabinoid molecules in HK-2 renal cells

1. Endogenous and synthetic cannabinoid molecules have been investigated as possible MDR-1/P-glycoprotein (P-gp) modulators in HK-2-immortalized renal cells, using calcein acetoxymethylester (calcein-AM) as a P-gp substrate. 2. Among the endocannabinoid molecules tested, anandamide (AEA), but not 2-...

詳細記述

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書誌詳細
主要な著者: Nieri, Paola, Romiti, Nadia, Adinolfi, Barbara, Chicca, Andrea, Massarelli, Ilaria, Chieli, Elisabetta
フォーマット: Artigo
言語:Inglês
出版事項: Nature Publishing Group 2006
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC1751877/
https://ncbi.nlm.nih.gov/pubmed/16715117
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0706778
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